Ceyone Life Sciences

CAS Number 202189-78-4
Category Second-Generation H1 Antihistamine
Final Application Antihistamine
Molecular Formula C28H37N3O3
Molecular Weight 463.61

Bilastine is a second-generation, non-sedating H1-receptor antagonist used to relieve symptoms of allergic rhinoconjunctivitis and chronic urticaria. Minimal CNS penetration gives it a favorable low-sedation profile compared with first-generation antihistamines, and it is typically dosed once daily.